PUBLICAÇÕES
SELECIONADAS

- Da Silva, Jaqueline; Gabriel-Costa, Daniele; Sudo, Roberto; Wang, Hao; Groban, Leanne; Ferraz, Emanuele; Nascimento, Jose; Fraga, Carlos A. M.; Barreiro, Eliezer; Zapata-Sudo, Gisele. Adenosine A2a Receptor Agonist Prevents Cardiac Remodeling And Dysfunction In Spontaneously Hypertensive Male Rats After Myocardial Infarction. Drug Design Development and Therapy, v. 11, p. 553-562, 2017. [Link]
- Betti, Andresa H.; Antonio, Camila B.; Pompeu, Thais E. T.; Martins, Thaise S.; Herzfeldt, Vivian; Stolz, Eveline D.; Fraga, Carlos A. M.; Barreiro, Eliezer; Noël, François; Rates, Stela M. K. LASSBio-1422: A New Molecular Scaffold With Efficacy In Animal Models Of Schizophrenia And Disorders Of Attention And Cognition. Behavioural Pharmacology, v. 28, p. 48-62, 2017. [Link]
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Ibiapino, Amanda Laura; De Figueiredo, Laysa Pires; Lima, Lídia Moreira; Barreiro, Eliezer J.; Punzo, Francesco; Ferreira, Fabio Furlan. Structural and Physicochemical Characterization Of Sulfonylhydrazone Derivatives Designed as Hypoglycemic Agents. New Journal Of Chemistry, v. 41, v. 6464-6474, 2017. [Link]
- De Figueiredo, Laysa P.; Ibiapino, Amanda L.; Do Amaral, Daniel N.; Ferraz, Letícia S.; Rodrigues, Tiago; Barreiro, Eliezer J.; Lima, Lídia M.; Ferreira, Fabio F. Structural Characterization And Cytotoxicity Studies of Different Forms of A Combretastatin A4 Analogue. Journal of Molecular Structure, v. 1147, p. 226-234, 2017. [Link]
- Bastos, Isadora T. S.; Costa, Fanny N.; Silva, Tiago F.; Barreiro, Eliezer J.; Lima, Lídia M.; Braz, Delson; Lombardo, Giuseppe M.; Punzo, Francesco; Ferreira, Fabio F.; Barroso, Regina C. A Combined Experimental and In Silico Characterization To Highlight Additional Structural Features And Properties Of A Potentially New Drug. Journal of Molecular Structure, v. 1146, p. 735-743, 2017. [Link]
- Frattani, Flávia S.; Lima, Lidia M.; Barreiro, Eliezer J.; Zingali, Russolina B. The Antithrombotic and Haemostatic Effects Of Lassbio-752: A Synthetic, Orally Active Compound in an Arterial and Venous Thrombosis Model in Rats. Journal of Pharmacy and Pharmacology, v. 69, p. 1374-1380, 2017. [Link]
- Do Amaral, Daniel; De Sá Alves, Fernando; Barreiro, Eliezer; Laufer, Stefan; Lima, Lídia. Multi-Gram Preparation Of 7-Nitroquinoxalin-2-Amine. Journal of The Brazilian Chemical Society, v. 28, p. 1874-1878, 2017. [Link]
- Alencar, Allan K. N.; Montes, Guilherme C.; Barreiro, Eliezer J.; Sudo, Roberto T.; Zapata-Sudo, Gisele. Adenosine Receptors as Drug Targets For Treatment of Pulmonary Arterial Hypertension. Frontiers in Pharmacology, v. 8, p. 858, 2017. [Link]
- Carvalho, Vinicius F.; Ferreira, Tatiana P. T.; De Arantes, Ana C. S.; Noël, François; Tesch, Roberta; Sant’Anna, Carlos M. R.; Barreiro, Eliezer J.; Fraga, Carlos A. M.; Rodrigues E Silva, Patrícia M.; Martins, Marco A. Lassbio-897 Reduces Lung Injury Induced by Silica Particles in Mice: Potential Interaction With The A2a Receptor. Frontiers in Pharmacology, V. 8, P. 778, 2017. [Link]
- Carvalho, Samir Aquino; Osorio, Luis Felipe Baumotte; Salomão, Kelly; De Castro, Solange Lisboa; Wardell, Solange M. S. V.; Wardell, James Lewis; Da Silva, Edson Ferreira; Fraga, Carlos A. M. Design, Synthesis, and Trypanocidal Activity pf Novel 5-nitroimidazolyl O-Benzyloxime Ethers. Journal of Heterocyclic Chemistry, v. 54, p. 3626-3631, 2017. [Link]
- Guerra, Fabiana Sélos; Oliveira, Ramon Guerra de; Fraga, Carlos Alberto Manssour; Mermelstein, Claudia Dos Santos; Fernandes, Patricia Dias. Rock Inhibition With Fasudil Induces Beta-Catenin Nuclear Translocation and Inhibits Cell Migration of MDA-MB 231 Human Breast Cancer Cells. Scientific Reports, v. 7, p. 13723, 2017. [Link]
- Elizondo-Jimenez, Silvia; Moreno-Herrera, Antonio; Reyes-Olivares, Rogelio; Dorantes-Gonzalez, Edith; Nogueda-Torres, Benjamín; De Oliveira, Eduardo; Romeiro, Nelilma; Lima, Lidia; Palos, Isidro; Rivera, Gildardo. Synthesis, Biological Evaluation and Molecular Docking of New Benzenesulfonylhydrazone as Potential Anti-Trypanosoma cruzi Agents. Medicinal Chemistry, v. 13, p. 149-158, 2017. [Link]
- Moraes, Barbra Sanches; Azeredo, Francine Johansson; Izoton, Jessica Cristina; Amaral, Marina; Barreiro, Eliezer; Freddo, Rodrigo José; Dalla Costa, Teresa; Lima, Lídia Moreira; Haas, Sandra Elisa. Leishmanicidal Candidate Lassbio-1736, a Cysteine Protease Inhibitor with Favorable Pharmacokinetics: Low Clearance And Good Distribution. Xenobiotica, 2017. [Link] (In press)
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Carneiro, Teiliane R.; Do Amaral, Daniel N.; Fokoue, Harold H.; Sant'Anna, Carlos M. R.; Porras, Maria; Pessoa, Cláudia; Oliveira, Augusto; Barreiro, Eliezer; Cavalcanti, Bruno; Lima, Lidia Moreira. Synthesis, Pharmacological Evaluation and Docking Study of a New Modulator of Microtubule Polymerization. Letters in Drug Design & Discovery, 2017. [Link] (In press)
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